Specificity protein 1-modulated superoxide dismutase 2 enhances temozolomide resistance in glioblastoma, which is independent of O6-methylguanine-DNA methyltransferase

Aug 20, 2017Redox biology

A protein that increases antioxidant enzyme levels may raise drug resistance in brain cancer, independent of a common DNA repair enzyme

AI simplified

Abstract

Increased expression of the protein Sp1 is associated with reduced levels of reactive oxygen species in temozolomide-resistant glioblastoma cells.

  • Temozolomide resistance in glioblastoma may occur independently of the DNA repair enzyme MGMT.
  • TMZ-resistant glioblastoma variants show elevated Sp1 expression and decreased reactive oxygen species accumulation after treatment.
  • The enzyme superoxide dismutase 2 (SOD2) is identified as a disease-related ROS scavenger that is co-expressed with Sp1 in resistant cells.
  • Sp1 acts as a key activator of the SOD2 gene, enhancing its expression.
  • Inhibition of Sp1 can reverse TMZ resistance and lower SOD2 levels in resistant glioblastoma cells.
  • This inhibition strategy improved survival rates in an animal model of glioblastoma.

AI simplified

Full Text

We can’t show the full text here under this license. Use the link below to read it at the source.

what lands in your inbox each week:

  • 📚7 fresh studies
  • 📝plain-language summaries
  • direct links to original studies
  • 🏅top journal indicators
  • 📅weekly delivery
  • 🧘‍♂️always free