A review of GLP‐1 receptor agonists in type 2 diabetes: A focus on the mechanism of action of once‐weekly agents

Sep 10, 2020Journal of clinical pharmacy and therapeutics

How once-weekly GLP-1 drugs work in type 2 diabetes

AI simplified

Abstract

Glucagon-like peptide-1 receptor agonists (GLP-1 RAs) may provide multi-factorial clinical benefits for people with type 2 diabetes (T2D).

  • GLP-1 RAs lower blood glucose through mechanisms such as enhancing insulin secretion and reducing glucagon release.
  • These medications can slow gastric emptying and promote feelings of fullness.
  • GLP-1 RAs may have positive effects on cardiovascular and renal health due to the presence of GLP-1 receptors in these organ systems.
  • Variations in the molecular size, structure, and duration of action among individual GLP-1 RAs lead to differences in their pharmacodynamics and clinical outcomes.
  • Pharmacists play a key role in medication management and should consider the specific mechanisms of action when advising on GLP-1 RA treatments.

AI simplified

Key numbers

−2.0 to −7.9 kg
Weight Reduction Range (Semaglutide)
Average body weight reductions in clinical studies with semaglutide.
−1.4 to −4.1 kg
Weight Reduction Range (Exenatide ER)
Average body weight reductions in clinical studies with exenatide ER.
26%
Risk Reduction in MACE (Semaglutide)
Reduced risk of MACE in high-risk T2D patients treated with semaglutide.

Full Text

We can’t show the full text here under this license. Use the link below to read it at the source.

what lands in your inbox each week:

  • 📚7 fresh studies
  • 📝plain-language summaries
  • direct links to original studies
  • 🏅top journal indicators
  • 📅weekly delivery
  • 🧘‍♂️always free